1
Tarek A Zeidan, Scott Duncan, Christopher P Hencken, Thomas Andrew Wynn, Carlos N Sanrame: Prodrugs of fumarates and their use in treating various diseases. Alkermes Pharma Ireland, Lathrop & Gage, Brian C Trinque, March 11, 2014: US08669281 (20 worldwide citation)

The present invention provides compounds of formula (I), wherein: R1 is unsubstituted C1-C6 alkyl; La is substituted or unsubstituted C1-C6 alkyl linker, substituted or unsubstituted C3-C10 carbocycle, substituted or unsubstituted heterocycle comprising one or two 5- or 6-member rings and 1-4 hetero ...


2
Tarek A Zeidan, Scott Duncan, Christopher P Hencken, Thomas Andrew Wynn, Carlos N Sanrame: Prodrugs of fumarates and their use in treating various diseases. Alkermes Pharma Ireland, Elmore Patent Law Group P C, Carolyn S Elmore, July 28, 2015: US09090558 (13 worldwide citation)

The present invention provides compounds of formula (I), wherein: R1 is unsubstituted C1-C6 alkyl; La is substituted or unsubstituted C1-C6 alkyl linker, substituted or unsubstituted C3-C10 carbocycle, substituted or unsubstituted heterocycle comprising one or two 5- or 6-member rings and 1-4 hetero ...


3

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5
Ratan K Chaudhuri, Krys Bojanowski: Compositions and methods for treating psoriasis. SYMBIONYX PHARMACEUTICALS, Edward K Welch II, IP&L Solutions, May 2, 2017: US09636321

Novel isohexides and pharmaceutical compositions containing the same as well as methods of using the same in the treatment of psoriasis.


6
PRODRUGS OF FUMARATES AND THEIR USE IN TREATING VARIOUS DISEASES. Alkermes Pharma Ireland, September 18, 2014: US20140275048-A1

The present invention provides compounds of formula (I), and pharmaceutical compositions thereof.


7
PRODRUGS OF FUMARATES AND THEIR USE IN TREATING VARIOUS DISEASES. September 18, 2014: US20140275205-A1

The present invention provides compounds of formula (I), wherein: R1 is unsubstituted C1-C6 alkyl; La is substituted or unsubstituted C1-C6 alkyl linker, substituted or unsubstituted C3-C10 carbocycle, substituted or unsubstituted heterocycle comprising one or two 5- or 6-member rings and 1-4 hetero ...


8
SULFONAMIDE AND SULFINAMIDE PRODRUGS OF FUMARATES AND THEIR USE IN TREATING VARIOUS DISEASES. August 27, 2015: US20150239829-A1

The present invention provides compounds and pharmaceutical compositions for treating neurological diseases such as multiple sclerosis.


9
PRODRUGS OF FUMARATES AND THEIR USE IN TREATING VARIOUS DISEASES. May 19, 2016: US20160137660-A1

The present invention provides compounds of formula (I), wherein: R1 is unsubstituted C1-C6 alkyl; La is substituted or unsubstituted C1-C6 alkyl linker, substituted or unsubstituted C3-C10 carbocycle, substituted or unsubstituted heterocycle comprising one or two 5- or 6-member rings and 1-4 hetero ...


10
PRODRUGS OF FUMARATES AND THEIR USE IN TREATING VARIOUS DISEASES. April 6, 2017: US20170095439-A1

The present invention provides compounds of formula (I), and pharmaceutical compositions thereof.