1
Metternich Rainer: Peptide boronic acid derivatives having protease inhibiting activity.. Sandoz, Sandoz, Sandoz, February 19, 1992: EP0471651-A2 (84 worldwide citation)

Borolysine peptidomimetics of formula I wherein W, Y, R4, R5, Q1 and Q2 are defined in claim 1 are potent thrombin inhibitors.


2

3
Cook Nigel Scott, Metternich Rainer, Tapparelli Carlo, Wienand Anette: Peptide boronic acid derivatives having protease inhibiting activity. Sandoz, Sandoz, Sandoz, December 27, 1995: EP0688336-A1

Peptidomimetics of formula (I), wherein W, Y, R4, R5, Q1 and Q2 are defined in claim 1 are potent thrombin inhibitors.