1
Setoi Hiroyuki, Ohkawa Takehiko, Zenkoh Tatsuya, Hemmi Keiji, Tanaka Horokazu: Benzamide derivatives and their use as vasopressin antagonists.. Fujisawa Pharmaceutical Co, October 19, 1994: EP0620216-A1 (58 worldwide citation)

A compound of the formula : wherein R is hydrogen or lower alkyl, R is hydrogen, lower alkyl, halo(lower)alkyl, halogen or lower alkoxy, R and R are each hydrogen, lower alkyl or taken together to form oxo, R is hydrogen, halogen, nitro, hydroxy, protected hydroxy, lower alkyl or lower alkoxy option ...


2
Hiroyuki Setoi, Takehiko Ohkawa, Tatsuya Zenkoh, Hitoshi Sawada, Kentaro Sato, Hirokazu Tanaka: Benzamide derivatives and their use as vasopressin antagonists. Fujisawa Pharmaceutical, Oblon Spivak McClelland Maier & Neustadt P C, April 25, 2000: US06054457 (25 worldwide citation)

This invention relates to new benzamide derivatives having a vasopressin antagonistic activity, etc, and represented by general formula (I): ##STR1## wherein R.sup.1 is aryl optionally substituted with lower alkoxy, etc., R.sup.2 is lower alkyl, etc.,


3
Setoi Hiroyuki, Ohkawa Takehiko, Zenkoh Tatsuya, Sawada Hitoshi, Sato Kentaro, Tanaka Hirokazu: Benzamide derivatives and their use as vasopressin antagonists. Fujisawa Pharmaceutical Co, April 1, 1998: EP0832061-A1 (1 worldwide citation)

This invention relates to new benzamide derivatives having a vasopressin antagonistic activity, etc., and represented by general formula (I), wherein R is aryl optionally substituted with lower alkoxy, etc., R is lower alkyl, etc., R is hydrogen, etc., R is lower alkoxy, etc., R is hydrogen, etc., A ...


4
Setoi Hiroyuki, Zenkoh Tatsuya, Sawada Hitoshi: Benzamide derivatives and their use as vasopressin antagonists. Fujisawa Pharmaceutical, liu yuanjin, September 9, 1998: CN96196175

This invention relates to new benzamide derivatives having a vasopressin antagonistic activity, etc, and represented by general formula (I), wherein R is aryl optionally substituted with lower alkoxy, etc, R is lower alkyl, etc, R is hydrogen, etc, R is lower alkoxy, etc, R is hydrogen, etc, A is NH ...


5
Setoi Hiroyuki, Ohkawa Takehiko, Zenkoh Tatsuya, Sawada Hitoshi, Sato Kentaro, Tanaka Hirokazu: Benzamide derivatives and their use as vasopressin antagonists. Fujisawa Pharmaceutical, Setoi Hiroyuki, Ohkawa Takehiko, Zenkoh Tatsuya, Sawada Hitoshi, Sato Kentaro, Tanaka Hirokazu, SEKI Hideo, December 27, 1996: WO/1996/041795

This invention relates to new benzamide derivatives having a vasopressin antagonistic activity, etc., and represented by general formula (I), wherein R?1¿ is aryl optionally substituted with lower alkoxy, etc., R?2¿ is lower alkyl, etc., R?3¿ is hydrogen, etc., R?4¿ is lower alkoxy, etc., R?5¿ is hy ...