1
Jean Luc Girardet, Yung Hyo Koh: 2-(5-bromo-4-(4-cyclopropylnaphthalen-1-yl)-4H-1,2,4-triazol-3-ylthio)acetic acid and methyl ester. Ardea Biosciences, Wilson Sonsini Goodrich & Rosati, August 23, 2011: US08003681 (17 worldwide citation)

A series of S-triazolyl α-mercaptoacetanilides having general structure (1) are provided, where Q is CO2H, CONR2, SO3H, or SO2NR2. The compounds inhibit several variants of the reverse transcriptase of HIV, and are useful in the treatment of HIV infections.


2
Jean Luc Girardet, Yung Hyo Koh: 2-(5-bromo-4-(4-cyclopropylnaphthalen-1-yl)-4h-1,2,4-triazol-3-ylthio)acetic acid and methyl ester. Wilson Sonsini Goodrich & Rosati, March 18, 2010: US20100069645-A1

A series of S-triazolyl α-mercaptoacetanilides having general structure (I) are provided, where Q is CO2H, CONR2, SO3H, or SO2NR2. The compounds inhibit several variants of the reverse transcriptase of HIV, and are useful in the treatment of HIV infections.


3
Jean Luc Girardet, Yung Hyo Koh: 2-(5-bromo-4-(4-cyclopropylnaphthalen-1-yl)-4h-1,2,4-triazol-3-ylthio)acetic acid and methyl ester. Ardea Biosciences, Wilson Sonsini Goodrich & Rosati, April 1, 2010: US20100081827-A1

A series of S-triazolyl α-mercaptoacetanilides having general structure (1) are provided, where Q is CO2H, CONR2. SO3H or SO2NR2. The compounds inhibit several variants of the reverse transcriptase of HIV, and are useful in the treatment of HIV infections.