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James Doherty
Dorn Conrad P, Finke Paul E, Maccoss Malcolm, Doherty James B, Shah Shrenik K, Hagmann William K: New substituted azetidinones as anti-inflammatory and antidegenerative agents.. Merck & Co, April 22, 1992: EP0481671-A1 (40 worldwide citation)

New substituted azetidinones of the general formula (A') which have been found to be potent elastase inhibitors and thereby useful anti-inflammatory and antidegenerative agents are described. e


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Eric First, M.D.
Eric R First: Methods for treating gluteal muscle. Allergan, Allergan, June 26, 2008: US20080152672-A1

Methods for treating a buttock deformity or for preventing development of a buttock deformity by local administration of a Clostridial toxin, such as a botulinum neurotoxin, to a buttock deformity or to the vicinity of a buttock deformity.


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Tammy Balzar
Sarah A Lemke, Scott W Wenzel, Tammy J Balzar: Skin cooling composition. Kimberly Clark Worldwide, Catherine E Wolf, April 30, 2009: US20090110656-A1

A cooling composition for application to the skin of a mammal, such as a human. The base of the composition is an interpenetrating polymer network, which may contain a thermo-responsive polymer. Having a Critical Temperature above an average core body temperature, the material may undergo a phase ch ...


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Handa Balraj Krishan, Machin Peter James, Martin Joseph Armstrong, Redshaw Sally, Thomas Gareth John: Amino acid derivatives.. Hoffmann La Roche, December 20, 1989: EP0346847-A2 (262 worldwide citation)

Compounds of the formula wherein R represents alkoxycarbonyl, aralkoxycarbonyl, alkanoyl, cycloalkylcarbonyl, aralkanoyl, aroyl, heterocyclylcarbonyl, alkylsulphonyl, arylsulphonyl, monoaralkylcarbamoyl, cinnamoyl or alpha -aralkoxycarbonylaminoalkanoyl and R represents hydrogen or R and R together ...


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Sigal Irving S, Huff Joel R, Darke Paul L, Vacca Joseph P, Young Steven D, Desolms S Jane, Thompson Wayne J, Lyle Terry A, Graham Samuel L, Ghosh Arun K: Hiv protease inhibitors useful for the treatment of aids.. Merck & Co, October 18, 1989: EP0337714-A2 (242 worldwide citation)

Compounds of the form A-G-B-B-J wherein A is an amine protecting group commonly employed in peptide synthesis, G a dipeptide isostere, B an amino acid or analog thereof, and J a small terminal group are described. These compounds are useful in the inhibition of HIV protease, the prevention or treatm ...


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Chakravarty Prasun K, Greenlee William J, Mantlo Nathan B, Patchett Arthur A, Walsh Thomas F: Substituted imidazo-fused 6-membered heterocycles as angiotensin ii antagonists.. Merck & Co, December 5, 1990: EP0400974-A2 (191 worldwide citation)

Substituted Imidazo-fused 6-membered heterocycles of structural formula: wherein A, B, C, and D are independently carbon atoms or nitrogen atoms are angiotensin II antagonists useful in the treatment of hypertension and congestive heart failure.


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Hunziker Ernst B: Kits and compositions for the treatment and repair of defects or lesions in cartilage or bone.. Shaw Robert F, March 10, 1993: EP0530804-A1 (187 worldwide citation)

Kits and compositions are provided for the treatment and repair of defects in the cartilage or bone of humans and other animals as in full-thickness defects in joints. A matrix having pores large enough to allow cells to populate the matrix and to form blood vessels is used to fill the defect in bon ...


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Patchett Arthur A, Harris Elbert E, Wyvratt Matthew J, Tristram Edward W: Carboxyalkyl dipeptide derivatives, process for preparing them and pharmaceutical composition containing them.. Merck & Co, June 25, 1980: EP0012401-A1 (181 worldwide citation)

Carboxyalkyl dipeptide derivatives and related compounds which are useful as antihypertensives, and having the formulae: wherein R and R are the same or different and are hydroxy, alkoxy, alkenoxy, dialkylamino alkoxy, acylamino alkoxy, acyloxy alkoxy, aryloxy, alkyloxy, substituted aryloxy or subst ...