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Wortmann Lars, Menzenbach Bernd, Kosemund Dirk, Frenzel Thomas, Schrey Anna Katharina, Kühne Ronald, Muhn Peter, Liesener Florian Peter, Koppitz Marcus: Arylmethylen substituted n-acyl-gamma-aminoalcohols. Bayer Schering Pharma Aktiengesellschaft, Wortmann Lars, Menzenbach Bernd, Kosemund Dirk, Frenzel Thomas, Schrey Anna Katharina, Kühne Ronald, Muhn Peter, Liesener Florian Peter, Koppitz Marcus, November 6, 2008: WO/2008/131972 (7 worldwide citation)

The present invention relates to arylmethylen substituted N-acyl-&ggr;-aminoalcohols of the general formula (I) in which Q, X, W, R1, R2, R3, R4 and R5 have the meaning as defined in the description. The Compounds according to the invention are effective FSH modulators and can be used for example fo ...


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Wortmann Lars, Menzenbach Bernd, Koppitz Marcus, Kosemund Dirk, Muhn Hans Peter, Schrey Anna, Kuehne Ronald, Frenzel Thomas, Liesener Florian Peter: Bicyclic acyltryptophanols. Bayer Schering Pharma Aktiengesellschaft, Wortmann Lars, Menzenbach Bernd, Koppitz Marcus, Kosemund Dirk, Muhn Hans Peter, Schrey Anna, Kuehne Ronald, Frenzel Thomas, Liesener Florian Peter, June 19, 2008: WO/2008/071455 (6 worldwide citation)

The present invention relates to acyltryptophanols of the general formula (I), in which Q, V, X, W, R1, R2, R3, R4, R5, R6, R7 and R8 have the meaning as defined in the description. The compounds according to the invention are effective FSH antagonists and can be used for example for fertility contr ...


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Wortmann Lars, Koppitz Marcus, Menzenbach Bernd, Kosemund Dirk, Schmees Norbert, Muhn Hans Peter, Frenzel Thomas, Liesener Florian Peter, Schrey Anna Katharina, Kühne Ronald: Arylmethylene substituted n-acyl-β-amino alcohols. Bayer Schering Pharma Aktiengesellschaft, Wortmann Lars, Koppitz Marcus, Menzenbach Bernd, Kosemund Dirk, Schmees Norbert, Muhn Hans Peter, Frenzel Thomas, Liesener Florian Peter, Schrey Anna Katharina, Kühne Ronald, January 29, 2009: WO/2009/013354 (5 worldwide citation)

The present invention relates to arylmethylene substituted N-Acyl-β-amino alcohols of the formula (I) : in which Y is selected from the aryl or heteroaryl groups: formula (II); and R1, R2, R3, R4, R5, Q, X and W have the meaning as defined in the description. The compounds according to the invention ...


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Wortmann Lars, Koppitz Marcus, Muhn Hans Peter, Frenzel Thomas, Liesener Florian Peter, Schrey Anna Katharina, Kühne Ronald: Cyanomethyl substituted n-acyl tryptamines. Bayer Schering Pharma Aktiengesellschaft, Wortmann Lars, Koppitz Marcus, Muhn Hans Peter, Frenzel Thomas, Liesener Florian Peter, Schrey Anna Katharina, Kühne Ronald, February 5, 2009: WO/2009/016253 (5 worldwide citation)

The present invention relates to cyanomethyl substituted N-acyl tryptamines of the formula (I) in which R1, R2, R3, R4, R5, Q, X and W have the meaning as defined in the description. The compounds according to the invention are effective FSH antagonists and can be used for example for fertility cont ...


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Wortmann Lars, Cleve Arwed, Muhn Hans Peter, Langer Gernot, Schrey Anna, Kühne Ronald, Menzenbach Bernd, Koppitz Marcus, Kosemund Dirk: Acyltryptophanols for fertility control. Bayer Schering Pharma Aktiengesellschaft, Wortmann Lars, Cleve Arwed, Muhn Hans Peter, Langer Gernot, Schrey Anna, Kühne Ronald, Menzenbach Bernd, Koppitz Marcus, Kosemund Dirk, February 15, 2007: WO/2007/017289 (5 worldwide citation)

The present patent application relates to acyltryptophanols of the general formula I, in which Q, X, Y, W, R1, R2, R3, R4, R5, R8 have the meanings stated in the description. The compounds according to the invention are effective FSH antagonists and can be used for example for fertility control in m ...


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Schulze Volker, Eis Knut, Wortmann Lars, Schwede Wolfgang, Siemeister Gerhard, Briem Hans, Schneider Herbert, Eberspächer Uwe, Hess Stumpp Holger: (De) Thiozolidinone, deren herstellung und verwendung als arzneimittel, (En) Thiozolidinones, production and use thereof as medicaments. Schering Aktiengesellschaft, Schulze Volker, Eis Knut, Wortmann Lars, Schwede Wolfgang, Siemeister Gerhard, Briem Hans, Schneider Herbert, Eberspächer Uwe, Hess Stumpp Holger, May 12, 2005: WO/2005/042505 (4 worldwide citation)

(EN) The invention relates to thiazolidinones of general formula ( I ), wherein Q, A, B, X, R1 and R2 have the meaning cited in the description, and the general formula (IA) wherein Q, A, B, X, R1 and R2a have the meaning cited in the description, to the production and use thereof as inhibitors of t ...


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KLAR Ulrich, WORTMANN Lars, KETTSCHAU Georg, PÜHLER Florian, LIENAU Philip, PETERSEN Kirstin, HÄGEBARTH Andrea, SÜLZLE Detlev: [fr] PYRROLOPYRIMIDINYLAMINOBENZOTHIAZOLONES SUBSTITUÉES COMME INHIBITEURS DE MKNK KINASE, [en] SUBSTITUTED PYRROLOPYRIMIDINYLAMINO-BENZOTHIAZOLONES AS MKNK KINASE INHIBITORS. BAYER PHARMA AKTIENGESELLSCHAFT, BIP PATENTS, March 27, 2014: WO/2014/044691 (3 worldwide citation)

[en] The present invention relates to substituted pyrrolopyrimidinylamino-benzothiazolone compounds of general formula I as described and defined herein, to methods of preparing said compounds, to intermediate compounds useful for preparing said compounds, to pharmaceutical compositions and combinat ...


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Wortmann Lars, Muhn Hans Peter, Menzenbach Bernd, Schrey Anna, Kuehne Ronald, Kosemund Dirk, Koppitz Marcus: 1,2-diarylacetylene derivatives of acyltryptophanols. Bayer Schering Pharma Aktiengesellschaft, Wortmann Lars, Muhn Hans Peter, Menzenbach Bernd, Schrey Anna, Kuehne Ronald, Kosemund Dirk, Koppitz Marcus, June 19, 2008: WO/2008/071453 (1 worldwide citation)

The present invention relates to acyltryptophanols of the general formula (I) in which Q, W, R1, R2, R3, R4, R5, R6, R7 and R8 have the meaning as defined in the description. The compounds according to the invention are effective FSH antagonists and can be used for example for fertility control in m ...