1
Guillemont Jerôme Emile Georges, Paugam Mikaël, Delest Bruno François Marie: Hiv inhibiting 5-amido substituted pyrimidines. Tibotec Pharmaceuticals, Guillemont Jerôme Emile Georges, Paugam Mikaël, Delest Bruno François Marie, WANTE Dirk, October 11, 2007: WO/2007/113254 (47 worldwide citation)

This invention concerns pyrimidine derivatives of formula having HIV (Human Immunodeficiency Virus) replication inhibiting properties, the preparation thereof and pharmaceutical compositions comprising these compounds.


2
Guillemont Jerôme Emile Georges, Paugam Mikaël, Delest Bruno François Marie, Heeres Jan, Lewi Paulus Joannes, Janssen Paul Adriaan Jan: Hiv inhibiting bicyclic pyrimidine derivatives. Tibotec Pharmaceuticals, Guillemont Jerôme Emile Georges, Paugam Mikaël, Delest Bruno François Marie, Heeres Jan, Lewi Paulus Joannes, Arts Frank Xavier Jozef Herwig, WANTE Dirk, May 4, 2006: WO/2006/045828 (46 worldwide citation)

HIV replication inhibitors of formula (I) N-oxides, pharmaceutically acceptable addition salts, quaternary amines or stereoisomeric forms thereof, wherein -a1=a2-a3=a4- is -CH=CH-CH=CH-, -N=CH-CH=CH-, -N=CH-N=CH-, -N=CH- CH=N-, -N=N-CH=CH-; -b1=b2-b3=b4- is -CH=CH-CH=CH-, -N=CH-CH=CH-, -N=CH-N=CH-, ...