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EMMANUEL MICHEL JOSE, GUO XIN, KIM JIN MI, LO HO YIN, NEMOTO PETER ALLEN, QIAN KEVIN CHUNGENG: INHIBITEURS DAZA-BENZIMIDAZOLONE CHYMASE, AZA-BENZIMIDAZOLONE CHYMASE INHIBITORS. BOEHRINGER INGELHEIM INTERNATIONAL, BOEHRINGER INGELHEIM INTERNATIONAL, FETHERSTONHAUGH & CO, September 13, 2016: CA2736522

Disclosed are small molecule inhibitors of the formula (I): and the pharmaceutical compositions thereof and processes of making the same. The compounds are useful in treating various diseases and conditions involving chymase.