1
Nagao Yoshihiro, Konno Fujiko, Kotake Jiro, Ishii Fumio, Honda Haruyoshi, Sato Susumu: Alpha-substituted phenylpropionic acid derivative and medicine containing the same. Ssp, March 24, 1999: EP0903343-A1 (50 worldwide citation)

Disclosed herein are an alpha -substituted phenylpropionic acid derivative represented by the following general formula (1): wherein W is a (substituted) lactam ring, A is an alkylene or alkyleneoxy group or the like, X is O, S, NH or CH2, Y is an amino, hydroxy or lower alkoxy group, R is H, alkyl ...


2
Konno Fujiko, Nakazawa Kyoko, Hirota Hiroyuki, Ishida Kazuya, Kaneko Yasushi, Okouchi Hisako: (Ja) 抗真菌活性を有する新規ピラゾール化合物, (En) Novel pyrazole compounds having antifungal activity. Ssp, Konno Fujiko, Nakazawa Kyoko, Hirota Hiroyuki, Ishida Kazuya, Kaneko Yasushi, Okouchi Hisako, THE PATENT CORPORATE BODY ARUGA PATENT OFFICE, April 22, 2004: WO/2004/033432 (15 worldwide citation)

(EN) A pyrazole compound represented by the following general formula (I) or its salt and a drug containing the same as the active ingredient: (I) wherein R1, R2, R3, R4 and R5 represent each a substituent; and X represents a methine group or a nitrogen atom. The above compound is useful as a preven ...


3
Okada Tomomi, Konno Fujiko, Kaihoh Terumitsu, Ishikawa Masago, Takahashi Yoshinori, Mizuno Hiroyuki, Honda Haruyoshi, Sato Susumu, Matsuda Hideaki: 4-(.alpha.-hydroxy-.alpha-aryl-alkylcarbonylamino)-piperidines for the treatment and prophylaxis of disorders of the urinary tract. Ss Pharmaceutical Co, January 2, 1997: EP0751127-A1 (9 worldwide citation)

Disclosed herein is a substituted piperidine derivative represented by the following general formula (1): wherein R means an aryl or heteroaryl group which may have at least one substituent, R denotes an alkyl, alkenyl or aralkyl group, R stands for a hydrogen atom or an alkyl group, and R is a hydr ...


4
Konno Fujiko, Kaneko Yasushi, Hoshikado Takeshi, Ishida Kazuya, Hasegawa Kazuki, Konagai Akihiro, Nishiwaki Shigeru, Namiki Chiaki: (Ja) 抗真菌活性を有する新規アゾール誘導体, (En) Novel azole derivative having antifungal activity. Hisamitsu Medical, Konno Fujiko, Kaneko Yasushi, Hoshikado Takeshi, Ishida Kazuya, Hasegawa Kazuki, Konagai Akihiro, Nishiwaki Shigeru, Namiki Chiaki, THE PATENT CORPORATE BODY ARUGA PATENT OFFICE, December 16, 2004: WO/2004/108684 (8 worldwide citation)

(EN) An azole derivative represented by the general formula (1): (wherein X represents nitrogen or CH; and Ar represents optionally substituted phenyl or an optionally substituted aromatic heterocyclic group) or a salt of the derivative; an intermediate for these; and a process for producing these c ...


5
Konno Fujiko, Umehara Norimitsu, Matsuda Hideaki, Katori Tatsuhiko: Quinoline derivatives.. Ss Pharmaceutical Co, March 29, 1989: EP0308897-A1 (7 worldwide citation)

A quinoline derivative represented by the following formula is disclosed. wherein R1 represents a hydrogen atom or an alkyl group which may contain a substituent and R2 represents an alkyl group which may contain a substituent, or R1 and R2 in combination with each other and with the adjacent nitrog ...


6
Konno Fujiko, Shibata Akihiro, Matsuda Hideaki, Asaoka Takemitsu, Kawahara Ryuichi, Taido Naokata, Kuraishi Tadayuki, Takeda Sunao: Quinolonecarboxylic acid derivative.. Ss Pharmaceutical Co, July 8, 1992: EP0493608-A1 (6 worldwide citation)

A quinolonecarboxylic acid derivative represented by general formula (1), its salt and an antibacterial agent containing the same as the active ingredient, wherein R represents hydrogen, alkyl, aralkyl or an ester residue which is hydrolyzable in vivo; R represents hydrogen or amino which may be sub ...


7
Kaiho Terumitsu, Takeda Sunao, Konno Fujiko, Shibata Akihiro, Matsumoto Masaru, Asaoka Takemitsu, Matsuda Hideaki, Kuraishi Tadayuki: 5-aminoquinolonecarboxylic acid derivative and antibacterial containing the same as active ingredient.. Ss Pharmaceutical Co, June 15, 1994: EP0601197-A1 (3 worldwide citation)

A 5-aminoquinolonecarboxylic acid derivative represented by general formula (1) or a salt thereof, and an antibacterial containing the same as the active ingredient, wherein R represents hydrogen, amino, C1-C5 linear or branched alkyl, or an alkylamino group having a C1-C5 linear or branched alkyl g ...


8
Konno Fujiko, Kaneko Yasushi, Hoshikado Takeshi, Ishida Kazuya, Hasegawa Kazuyoshi, Konagai Akihiro, Nishiwaki Shigeru, Namiki Chiaki: New azole derivative with antimycotic activity. Ss Pharmaceut, December 24, 2004: JP2004-359646 (1 worldwide citation)

PROBLEM TO BE SOLVED: To provide a new azole derivative with high safety, having antimycotic activity effective in deep mycosis and superficial mycosis.SOLUTION: The azole derivative is represented by general formula (1) (wherein X is N or CH. Ar is a phenyl group which may have a substituent or an ...


9
Konno Fujiko, Nagao Yoshihiro, Isomae Kazuo, Ohtsuka Mari, Takahashi Yoshiyuki, Ishii Fumio, Hirota Hiroyuki, Takeda Sunao, Kawamoto Noriyuki, Honda Haruyoshi, Sato Susumu: Imidazole derivatives or salts thereof and drugs containing the derivatives or the salts. Ssp, March 26, 2003: EP1295880-A1

The invention is directed to an imidazole derivative represented by formula (1): wherein each of R and R represents an aryl group, a heteroaryl group, etc.; each of A, X, and X represents N or CH; each of Y and Z represents O, S, etc.; each of R, R, and R represents a hydrogen atom, an alkyl group, ...


10
Ishii Fumio, Honda Haruyoshi, Konno Fujiko, Okada Tomomi, Kaihoh Terumitsu, Nagao Yoshihiro, Sato Susumu, Matsuda Hideaki: Chromene derivatives and salts thereof, and pharmaceuticals containing the same. Ssp, April 7, 1999: EP0906910-A1

Disclosed are chromene derivatives represented by the following formula: wherein Rs represent alkyl, alkoxy or like groups, R represents a hydrogen atom or an alkyl group, R represents a substituted or unsubstituted phenyl, naphthyl or heterocyclic group, and m stands for an integer of from 0 to 4, ...



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