1
Bela Kiss
János Galambos, Katalin Nógrádi, Éva Ágainé Csongor, György Miklós Keserü, István Vágó, György Domány, Béla Kiss, István Gyertyán, István Laszlovszky, Judit Laszy: Sulfonamide derivatives as D3-receptor ligands. Richter Gedeon Vegyeszeti Gyar Rt, Sterne Kessler Goldstein & Fox P L L C, January 6, 2009: US07473692

The present invention relates to new D3 dopamine receptor subtype selectice ligands of formula (I) to pharmacological compositions containing the same and to their use in therapy and/or prevention of psychoses (e.g. schizophrenia, schizo-affective disorders, etc), drug (e.g. alcohol, cocaine and nic ...


2
Gyorgy Domány, Csilla Horváth, Gizella Bartáné Szalai, József Nagy, Sándor Kolok, Éva Kovácsné Bozó, István Borza, István Vágó, Attila Bielik, Györgyi Ignáczné Szendrei, György Keserü, Sándor Farkas: Piperidine derivatives as NMDA receptor antagonists. Gedeon Richter Vegyeszeti Gyar RT, Rakoczy Molino Mazzochi Siwik, October 14, 2008: US07435744 (3 worldwide citation)

The present invention relates to a compound of formula (I): wherein: V and U are hydrogen, halogen, C1-C4 alkylamino, or together form a group that contains one or more heteroatoms, and that taken together with one or more: (a) hydrogen atoms; (b) carbon atoms; (c) —CH═ groups; (d) —CH2— groups; or ...