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Paul L Feldman, David Kendall Jung, Istvan Kaldor, Gregory J Pacofsky, Jeffrey A Stafford, Jeffrey H Tidwell: Short-acting benzodiazepines. CeNeS, Peter F Corless, Edwards Angell Palmer & Dodge, January 9, 2007: US07160880 (10 worldwide citation)

The present invention provides a compound of formula (I): wherein all variables are as defined herein, pharmaceutical formulations containing the same, processes for preparing the same and their use therapy.


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Paul L Feldman, David Kendall Jung, Istvan Kaldor, Gregory J Pacofsky, Jeffrey A Stafford, Jeffrey H Tidwell: Short-acting benzodiazepines. CeNes, Edwards Angell Palmer & Dodge, Peter F Corless, February 3, 2009: US07485635 (8 worldwide citation)

The present invention provides a compound of formula (I): wherein all variables are as defined herein, pharmaceutical formulations containing the same, processes for preparing the same and their use therapy.


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Paul L Feldman, David Kendall Jung, Istvan Kaldor, Gregory J Pacofsky, Jeffrey A Stafford, Jeffrey H Tidwell: Short-acting benzodiazepines. CeNes, Peter F Corless, Edwards Angell Palmer & Dodge, January 6, 2009: US07473689 (7 worldwide citation)

The present invention provides a compound of formula (I): wherein all variables are as defined herein, pharmaceutical formulations containing the same, processes for preparing the same and their use therapy.


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Paul L Feldman, David Kendall Jung, Istvan Kaldor, Gregory J Pacofsky, Jeffrey A Stafford, Jeffrey H Tidwell: Short-acting benzodiazepines. CeNeS, Peter F Corless, Edwards Angell Palmer & Dodge, October 14, 2008: US07435730 (7 worldwide citation)

The present invention provides a compound of formula (I): wherein all variables are as defined herein, pharmaceutical formulations containing the same, processes for preparing the same and their use therapy.


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Paul L Feldman, David Kendall Jung, Istvan Kaldor, Gregory J Pacofsky, Jeffrey A Stafford, Jeffrey H Tidwell: Short-acting benzodiazepines. CeNes, Peter F Corless, Edwards Angell Palmer & Dodge, May 5, 2009: US07528127 (7 worldwide citation)

It has now been found that compounds of the present invention as described in Benzodiazepine derivatives of Formula (I) containing a carboxylic ester moiety and thereby capable of being inactivated by nonspecific tissue esterases in an organ-independent elimination mechanism and thereby providing a ...


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Michael John Alberti, Ian Robert Baldwin, Mui Cheung, Stuart Cockerill, Stephen Flack, Philip Anthony Harris, David Kendall Jung, Gregory Peckham, Michael Robert Peel, Jennifer Gabriel Badiang, Kirk Stevens, James Marvin Veal: Fused pyrazole derivatives being protein kinase inhibitors. Glaxo Group, Lorie Ann Morgan, January 23, 2007: US07166597 (6 worldwide citation)

Compounds of Formula (I): salts or solvates or physiologically functional derivatives thereof, wherein Z is CH or N, and R1, R2, and R4 are various substituent groups, are protein kinase inhibitors


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Jennifer G Badiang, Scott Howard Dickerson, Philip Anthony Harris, David Kendall Jung, Michael Robert Peel, Michael John Reno, Tara Renae Rheault, Kirk Lawrence Stevens, Francis Xavier Tavares, James Marvin Veal: Pyrazolopyridazine derivatives. SmithKline Beecham Corporation, John L Lemanowicz, Kathryn L Coulter, October 9, 2007: US07279473 (2 worldwide citation)

Fused pyradazine derivatives which are usefule as CDK inhibitors are described herein. The described invention alos includes methods of making such fused pyradazine derivatives as wells as methods of using the same in the treatment of hyperproliferative diseases.


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Michael John Alberti, Stanley D Chamberlain, Mui Cheung, Kristjan Gudmundsson, Philip Anthony Harris, Brian A Johns, David Kendall Jung, Michael Robert Peel, Jennifer Badiang Stanford: Pyrazolopyridines, process for their preparation and use as therapeutic compounds. SmithKline Beecham Corporation, Lorie Ann Morgan, September 19, 2006: US07109209 (1 worldwide citation)

The present invention provides compounds of formula (I): wherein all variables are as defined herein, pharmaceutical compositions containing the same, processes for preparing the same and their use as pharmaceutical agents.