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Guillemont Jerome Emile George, Palandjian Patrice, de Jonge Marc Rene, Koymans Lucien Maria Henricus, Vinkers Hendrik Maarten, Daeyaert Frederik Frans Desire, Heeres Jan, Van Aken Koen Jeanne Alfons, Lewi Paulus Joannes, Janssen Paul Adriaan Jan: Hiv inhibiting pyrimidines derivatives. Janssen Pharmaceutica, May 19, 2004: EP1419152-A1 (2 worldwide citation)

This invention concerns HIV replication inhibitors of formula (I) the N -oxides, the pharmaceutically acceptable addition salts, the quaternary amines and the stereochemically isomeric forms thereof, wherein the ring containing -a=a-a=a- and -b=b-b=b- represents phenyl, pyridyl, pyrimidinyl, pirazin ...


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Buijnsters Peter Jacobus Johan, Daeyaert Frederik Frans Desire, Embrechts Werner Constant Joha, Freyne Eddy Jean Edgard, Geerts Hugo Alfons Gabriel, Heeres Jan, Janssen Paul Adriaan Jan, Jonge Marc Rene de, Koymans Lucien Maria Henricus, Kukla Michael Joseph, Lewi Paulus Joannes, Ludovici Donald William, Mercken Marc Hubert, Nuydens Rony Maria, Willems Marc: Aminobenzamide derivatives as glycogen synthase kinase 3 beta inhibitors. Janssen Pharmaceutica, guan lixin tan mengsheng, November 30, 2005: CN02821916 (1 worldwide citation)

This invention concerns a compound of formula (I),a N-oxide, a pharmaceutically acceptable addition salt, a quaternary amine and a stereochemically isomeric form thereof, wherein ring A represents a 6-membered heterocycle; R is hydrogen; aryl; formyl; C1-6alkylcarbonyl; optionally substituted C1-6al ...


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GUILLEMONT JEROME EMILE GEORGES, PALANDIJAN PATRICE, DE JONGE MARC RENE, KOYMANS LUCIEN MARIA HENRICUS, VINKERS HENDRIK MAARTEN, DAEYAERT FREDERIK FRANS DESIRE, HEERES JAN, VAN AKEN KOEN JEANNE ALFONS, LEWI PAULUS JOANNES, JANSSEN PAUL ADRIAAN JAN: [fr] Derivés dune pyrimidine en tant quinhibiteur du VIH, [de] HIV hemmende Pyrimidine Derivate, [en] HIV inhibiting pyrimidines derivatives. Janssen Pharmaceutica, March 23, 2011: EP2298761-A1

[en] This invention concerns HIV replication inhibitors of formula the N -oxides, the pharmaceutically acceptable addition salts, the quaternary amines and the stereochemically isomeric forms thereof, wherein the ring containing -a 1 =a 2 -a 3 =a 4 - and -b 1 =b 2 -b 3 =b 4 - represents phenyl, pyri ...


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Daeyaert Frederik Frans Desire, de Corte Bart, de Jonge Marc Rene, Heeres Jan, Ho Chih Yung, Janssen Paul Adriaan Jan, Kavash Robert W, Koymans Lucien Maria Henricus, Kukla Michael Joseph, Ludovici Donald William: Derives de 1,3,5-triazine trisubstitues pour le traitement dinfections a vih, Trisubstituted 1,3,5-triazine derivatives for treatment of hiv infections. Janssen Pharmaceutica, Janssen Pharmaceutica, GOWLING LAFLEUR HENDERSON, May 12, 2009: CA2324921

This invention concerns the use of the compounds of formula (I) the N-oxides, the pharmaceutically acceptable addition salts and the stereochemically isomeric forms thereof, wherein A is CH, CR4 or N; n is 0, 1, 2, 3 or 4; R1 and R2 are each independently selected from hydrogen, hydroxy, C1-12alkyl, ...