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BUCKMAN BRAD O, EMAYAN KUMAR, ISLAM IMADUL, MAY KAREN, BRYANT JUDI, MOHAN RAJU, WEST CHRISTOPHER L, YUAN SHENDONG: [fr] Dérivés de lacid phosphonic comme inhibiteurs de Plasma Carboxypeptidase B, [de] Phosphonsäure Derivaten als Plasma Carboxypeptidase B Inhibitoren, [en] Phosphonic acid as Plasma Carboxypeptidase B Inhibitors. BAYER SCHERING PHARMA, July 7, 2010: EP2204373-A1

[en] Compounds of the following formula (II), for example: wherein R 1 , R 2 , R 3 , and R 4 are described herein, are useful as inhibitors of plasma carboxypeptidase B. Pharmaceutical compositions containing these compounds, methods of using these compounds as antithrombotic agents and processes fo ...


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Bryant Judi, Buckman Brad, Islam Imadul, Mohan Raju, Morrissey Michael, Wei Guo Ping, Xu Wei, Yuan Shendong: Composes de 2-aminocarbonyl-quinoline utilises en tant quantagonistes du recepteur de ladenosine diphosphate des plaquettes, 2-aminocarbonyl-quinoline compounds as platelet adenosine diphosphate receptor antagonists. Schering Aktiengesellschaft, Bayer Schering Pharma Aktiengesellschaft, Marks & Clerk, May 31, 2011: CA2507657

Compounds of formula (I), where m, n, R1, R2, R3, R4 and R6 are described herein, are useful as inhibitors of platelet adenosine diphosphate. Pharmaceutical compositions containing these compounds, methods of using these compounds as antithrombotic agents and processes for synthesizing these compoun ...


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Bauman John G, Buckman Brad O, Ghannam Ameen F, Hesselgesser Joseph E, Horuk Richard, Islam Imadul, Liang Meina, May Karen B, Monahan Sean D, Morissey Michael M, Ng Howard P, Wei Guo Ping, Xu Wei, Zheng Wei, Shaw Kenneth J, Zuchun Zhao: Derives de piperazine et leur utilisation en tant quagents anti-inflammatoires, Piperazine derivatives and their use as anti-inflammatory agents. Schering Aktiengesellschaft, Schering Aktiengesellschaft, MARKS & CLERK, December 17, 1998: CA2293382

The invention is directed to acyl piperazine derivatiaves of formula Ia (see formula Ia) which are useful as anti-inflammatory agents. This invention is also directed to pharmaceutical compositions containing the compounds of the invention, and methods of using the compounds to treat inflammatory di ...


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Buckman Brad O, Davey David D, Guilford William J, Morrissey Michael M, Ng Howard P, Phillips Gary B, Wu Shung C, Xu Wei: Derives de benzamidine et utilisation de ces derives en tant quanticoagulants, Benzamidine derivatives their preparation and their use as anti-coagulants. Berlex Laboratories, Berlex Laboratories, BERESKIN & PARR, September 19, 1996: CA2214685

This invention is directed to benzamidine derivatives which are useful as anti-coagulants. This invention is also directed to pharmaceutical compositions containing the compounds of the invention, and methods of using the compounds to treat disease-states characterized by thrombotic activity. Accord ...


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Buckman Brad O, Emayan Kumar, Islam Imadul, May Karen, Bryant Judi, Mohan Raju, West Christopher, Yuan Shendong: Plasma carboxypeptidase b inhibitors. Schering, January 19, 2005: EP1497300-A2

Compounds of the following formula (I), for example: (1), wherein R, R, R, and R are described herein, are useful as inhibitors of plasma carboxypeptidase B. Pharmaceutical compositions containing these compounds, methods of using these compounds as antithrombotic agents and processes for synthesizi ...


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