1
Brown Matthew Lee, Cheung Mui, Dickerson Scott Howard, Gauthier Cassandra, Harris Philip Anthony, Hunter Robert Neil Iii, Pacofsky Gregory, Peel Michael Robert, Stafford Jeffrey Alan: Chemical compounds. Smithkline Beecham Corporation, Brown Matthew Lee, Cheung Mui, Dickerson Scott Howard, Gauthier Cassandra, Harris Philip Anthony, Hunter Robert Neil Iii, Pacofsky Gregory, Peel Michael Robert, Stafford Jeffrey Alan, LEVY David J, April 22, 2004: WO/2004/032882 (14 worldwide citation)

Oxazole derivatives, which are useful as VEGFR2, CDK2, and CDK4 inhibitors are described herein. The described invention also includes methods of making such oxazole derivatives as well as methods of using the same in the treatment of hyperproliferative diseases.


2

3

4
BROWN MATTHEW LEE, HOLZHAUSEN FRANZ VON, RAWLINSON PETER DORE, SAMPSON NICHOLAS JOHN, ECKERT MICHAEL JAMES, LEMIRE DAVID, VOLLMER AXEL BORIS: [fr] Porte de véhicule articulée double et procédé de commande associé, [de] Fahrzeugtür mit doppeltem Scharnier und Verfahren zur Steuerung davon, [en] Dual hinged vehicle door and method of controlling same. TESLA MOTORS, April 24, 2013: EP2583848-A2 (9 worldwide citation)

[en] A dual hinged door assembly for a vehicle is provided, the assembly including an upper door portion that pivots about a primary axis formed by its juncture with a structural member in the roof, and a lower door portion that pivots about a secondary axis formed by its juncture with the upper doo ...


5
Brown Matthew Lee, Cheung Mui, Dickerson Scott Howard, Gauthier Cassandra, Harris Philip Anthony, Hunter Robert Neil, Pacofsky Gregory, Peel Michael Robert, Stafford Jeffrey Alan: Chemical compounds. Smithkline Beecham, July 13, 2005: EP1551813-A2

Oxazole derivatives, which are useful as VEGFR2, CDK2, and CDK4 inhibitors are described herein. The described invention also includes methods of making such oxazole derivatives as well as methods of using the same in the treatment of hyperproliferative diseases.


6

7
Brown Matthew Lee, Cheung Mui, Dickerson Scott Howard, Drewry David Harold, Lackey Karen Elizabeth, Peat Andrew James, Thomson Stephen Andrew, Veal James Marvin, Wilson Jayme Lyn Roark: Pyrazolopyrimidines as kinase inhibitors. Smithkline Beecham, June 1, 2005: EP1534389-A2

The present invention relates to inhibitors of the kina ses GSK3 OR TIE2, and more particularly to pyrazolopyrimidine compounds useful as kinase inhibitors.