1
Ninkovic Sacha, Bennett Michael John, Rui Eugene Yuanjin, Wang Fen, Benedict Suzanne Pritchett, Teng Min, Wang Yong, Zhu Jinjiang: Diazepinoindole derivatives as kinase inhibitors. Pfizer, Ninkovic Sacha, Bennett Michael John, Rui Eugene Yuanjin, Wang Fen, Benedict Suzanne Pritchett, Teng Min, Wang Yong, Zhu Jinjiang, LUMB J Trevor, July 29, 2004: WO/2004/063198 (5 worldwide citation)

Protein kinase, such as CHK-1, inhibiting tricyclic compounds of the following formula (wherein R2, R3 and R4 are as defined in the specification) pharmaceutical compositions containing effective amounts of said compounds or their salts are useful as a single agent or in combination with an anti-neo ...


2
Chu Shao Song, Alegria Larry Andrew, Bender Steven Lee, Benedict Suzanne Pritchett, Borchardt Allen J, Kania Robert Steven, Nambu Mitchell David, Tempczyk Russell Anna Maria, Sarshar Sepehr, Bhumralkar Dilip, Peng Zhengwei, Yang Yi Michelle: Diaminothiazoles and their use for inhibiting protein kinases. Agouron Pharmaceuticals, PINO Mark J, December 14, 2000: WO/2000/075120 (4 worldwide citation)

Diaminothiazole compounds of formula (I) that modulate and/or inhibit the activity of certain protein kinases are described. These compounds and pharmaceutical compositions containing them are capable of mediating tyrosine kinase signal transduction in order to modulate and/or inhibit unwanted cell ...


3

4

5
Chu Shao Song, Alegria Larry Andrew, Bender Steven Lee, Benedict Suzanne Pritchett, Borchardt Allen J, Kania Robert Steven, Nambu Mitchell David, Tempczyk Russell Anna Maria, Sarshar Sepehr, Bhumralkar Dilip, Zhengwei Peng, Yang Yi Michelle: Diaminothiazoles and their use for inhibiting protein kinases. Agouron Pharma, February 27, 2002: EP1181283-A1

Diaminothiazole compounds of formula (I) that modulate and/or inhibit the activity of certain protein kinases are described. These compounds and pharmaceutical compositions containing them are capable of mediating tyrosine kinase signal transduction in order to modulate and/or inhibit unwanted cell ...


6
Nincovic Sacha, Bennett Michael John, Rui Eugene Yuanjin, Wang Fen, Benedict Suzanne Pritchett, Teng Min, Wang Yong, Zhu Jinjiang: Diazepinoindole derivatives as kinase inhibitors. Pfizer, September 21, 2005: KR1020057012806

Protein kinase, such as CHK-1, inhibiting tricyclic compounds of the following formula (wherein R2, R 3 and R4 are as defined in the specification) pharmaceutical compositions containing effective amounts of said compounds or their salts are useful as a single agent or in combination with an anti-ne ...


7
Chu Shao Song, Alegria Larry Andrew, Bender Steven Lee, Benedict Suzanne Pritchett, Borchardt Allen J, Kania Robert Steven, Nambu Michell David, Sarshar Sepehr, Tempczyk Russell Anna Maria, Bhumralkar Dilip, Zhengwei Peng, Yang Yi Michelle: Diaminothiazoles and their use for inhibiting protein kinases. Agouron Pharmaceuticals, February 27, 2002: KR1020017015384

Diaminothiazole compounds of formula (I) that modulate and/or inhibit the activity of certain protein kinases are described. These compounds and pharmaceutical compositions containing them are capable of mediating tyrosine kinase signal transduction in order to modulate and/or inhibit unwanted cell ...


8