1
Charles D Jones: Antiestrogenic and antiandrugenic benzothiophenes. Eli Lilly and Company, Joseph A Jones, Arthur R Whale, November 29, 1983: US04418068 (396 worldwide citation)

6-Hydroxy-2-(4-hydroxyphenyl)-3-[4-(2-piperidinoethoxy)benzoyl]benzo[b]thio phene, its ethers and esters, and the physiologically acceptable acid addition salts thereof, are valuable antiestrogens and antiendrogens.


2
C David Jones, Tulio Suarez: 2-Phenyl-3-aroylbenzothiophenes useful as antifertility agents. Eli Lilly and Company, William C Martens Jr, Arthur R Whale, January 9, 1979: US04133814 (352 worldwide citation)

Derivatives of 2-phenyl-3-aroylbenzothiophenes and 2-phenyl-3-aroylbenzothiophene-1-oxides are useful as antifertility agents. Certain of these compounds also are useful in suppressing the growth of mammary tumors.


3
Robert M Morris: Magnetically-localizable, biodegradable lipid microspheres. Eli Lilly and Company, James L Rowe, Arthur R Whale, May 25, 1982: US04331654 (296 worldwide citation)

Drug carrier formulation consisting of magnetically-localizable, biodegradable lipid microspheres.


4
Mary K Peters: Synthesis of acylated benzothiophenes. Eli Lilly and Company, Joseph A Jones, Arthur R Whale, April 19, 1983: US04380635 (237 worldwide citation)

A group of 6-hydroxy-2-(4-hydroxyphenyl)-3-[4-(2-aminoethoxy)benzoyl]benzo[b]thiophen es are prepared by acylation of a methyl-protected starting compound followed by demethylation in a single reaction mixture.


5
Nelson H Ludwig, Earl E Ose: Controlled release formulations and method of treatment. Eli Lilly and Company, Charles W Ashbrook, Arthur R Whale, October 6, 1981: US04293539 (148 worldwide citation)

Controlled release formulations useful in the prolonged treatment and control of microbial infections in animals are comprised of a microbial agent intimately dispersed throughout a copolymer derived from lactic acid and glycolic acid. A method for providing protection to animals for extended period ...


6
Bryan B Molloy, Klaus K Schmiegel: Arloxyphenylpropylamines. Eli Lilly and Company, James L Rowe, Arthur R Whale, February 2, 1982: US04314081 (121 worldwide citation)

3-Aryloxy-3-phenylpropylamines and acid additions salts thereof, useful as psychotropic agents, particularly as anti-depressants.


7
Robert S Nevin: Polymerization process and product. Eli Lilly and Company, Charles W Ashbrook, Arthur R Whale, June 16, 1981: US04273920 (108 worldwide citation)

Lactic-glycolic copolymers having molecular weights of about 6000 to about 35000 are prepared by condensation of lactic acid and glycolic acid in the presence of readily removable strong acid ion-exchange resins.


8
Tulio Suarez, C David Jones: Antifertility compounds. Eli Lilly and Company, William C Martens Jr, Arthur R Whale, October 28, 1980: US04230862 (104 worldwide citation)

Derivatives of 3-phenyl-4-aroyl-1,2-dihydronaphthalenes and 1-aroyl-2-phenylnaphthalenes are useful both as antifertility agents and in suppressing the growth of mammary tumors.


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Michele C Smith, Charles Pidgeon: Process for purifying proteins and compounds useful in such process. Eli Lilly and Company, William C Martens, Arthur R Whale, February 11, 1986: US04569794 (76 worldwide citation)

This invention describes a process for separating a biologically active polypeptide or protein in the form of its precursor from a mixture containing said precursor and impurities, which comprises contacting said precursor with a resin containing immobilized metal ions, said precursor comprising the ...