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Abdul B N Luheshi, Robert K Smalley, Peter D Kennewell, Robert Westwood: Process for the preparation of azabicyclo compounds. Roussel Uclaf, Bierman and Muserlian, February 4, 1992: US05086170 (368 worldwide citation)

A compound selected from the group consisting of a compound of the formula ##STR1## wherein R.sub.1 and R.sub.2 are individually selected from the group consisting of hydrogen, alkyl and hydroxyalkyl of 1 to 5 carbon atoms and amino, n is an integer from 1 to 3, X and X.sub.1 are individually select ...


2
Fernand Labrie, Jean Pierre Raynaud: Treatment method. Roussel Uclaf, Charles A Muserlian, September 18, 1984: US04472382 (87 worldwide citation)

A novel method of treating prostate adenocarcinoma, prostate benign hypertrophia, endometriosis, dysmenorrhea, hirsuitism, hormono-dependent mammary tumors, treatment and prevention of precocious puberty, induction of a retardation of the appearance of puberty and treatment of acne of mammals compri ...


3
Rene Heymes, Andre Lutz: 3-Acetoxymethyl-7-(iminoacetamido)-cephalosporanic acid derivatives. Roussel Uclaf, Hammond & Littell, May 1, 1979: US04152432 (72 worldwide citation)

Compounds of the formula ##STR1## wherein R is selected from the group consisting of hydrogen and groups easily removable by acid hydrolysis or hydrogenolysis, R' is selected from the group consisting of hydrogen, alkyl of 1 to 4 carbon atoms, alkenyl and alkynyl of 2 to 4 carbon atoms and groups ea ...


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Paul Zeitoun, Patrick Brisard: Compressed tablets for disintegration in the colon comprising an active ingredient containing nucleus coated with a first layer containing microcrystalline cellulose which is coated with an enteric organic polymer coating. Roussel UCLAF, Bacon & Thomas, February 21, 1984: US04432966 (70 worldwide citation)

Coated compressed tablets for oral administration are disclosed which substantially desintegrate specifically at the level of the colon. The tablets comprise a compressed center piece containing an active agent which center piece is coated by a first coating layer which is comprised of a mixture of ...


6
Jacques Perronnet, Pierre Girault, Claude Bonne: 1-(3-Trifluoromethyl-4-nitrophenyl)-4,4-dimethyl imidazolidines. Roussel Uclaf, Hammond & Littell, June 27, 1978: US04097578 (66 worldwide citation)

Imidazolidines of the formula ##STR1## wherein X is selected from the group consisting of oxygen and amine which inhibit the effects of androgens on peripheric receptors without interfering with normal hypophysial functions.


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Teutsch Jean Georges, Costerousse Germain, Philibert Daniel, Deraert Roger: Steroid derivatives substituted in the 11-beta position, process for their preparation, their utilization as medicaments and compositions containing them.. Roussel Uclaf, August 4, 1982: EP0057115-A2 (65 worldwide citation)

L'invention concerne les composés (I'): où R1 est un radical organique (1-18c), contenant un azote, un phosphore ou un silicium, R2 un radical hydrocarboné (1-8c), X le reste d'un cycle pentagonal ou hexagonal éventuellement substitué et insaturé C=A un groupe oxo libre ou bloqué ou un C=N-OH, C=N-O ...


8
Martine Gaillard Kelly, Francois Goubet, Daniel Philibert, Jean Georges Teutsch: Phenylimidazolidines having antiandrogenic activity. Roussel Uclaf, Bierman and Muserlian, May 2, 1995: US05411981 (63 worldwide citation)

A compound of the formula ##STR1## wherein R.sub.1 is --CN, --NO.sub.2 or halogen, R.sub.2 is --CF.sub.3 or halogen, --A-B-- is of ##STR2## X is --O-- or --S--, R.sub.3 is hydrogen, alkyl, alkenyl or alkynyl of up to 12 carbon atoms, aryl and aralkyl of up to 12 carbon atoms, all optionally substitu ...


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Constantin Agouridas, Yannick Benedetti, Jean Francois Chantot, Alexis Denis, Claude Fromentin, Odile Le Martret: Erythromycin compounds. Roussel UCLAF, Bierman and Muserlian, August 22, 1995: US05444051 (61 worldwide citation)

Compounds of the formula ##STR1## wherein X and X' form C.dbd.O or C.dbd.NOR, R is selected from the group consisting of hydrogen, heterocycle, alkyl, alkenyl, alkynyl, all optionally substituted,


10
Andre Allais, Francois Clemence, Roger Deraedt, Odile Le Martret: Quinoline-3-carboxamides. Roussel Uclaf, Hammond & Littell, August 15, 1978: US04107310 (56 worldwide citation)

Novel quinoline-3-carboxamides of the formula ##STR1## wherein R.sub.1 is in the 5,6,7 or 8-position and is selected from the group consisting of hydrogen, halogen, --CF.sub.3, --OCF.sub.3, --SCF.sub.3, straight chain alkyl of 1 to 4 carbon atoms, branched alkyl of 3 to 5 carbon atoms and alkoxy of ...



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