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Tamaki Kazuhiko, Yamaguchi Takahiro, Oda Kozo, Terasaka Naoki, Nakai Daisuke, Nakadai Masakazu: (Ja) 2以上の置換基を有するベンゼン化合物, (En) Benzene compound having 2 or more substituents. Daiichi Sankyo Company, Tamaki Kazuhiko, Yamaguchi Takahiro, Oda Kozo, Terasaka Naoki, Nakai Daisuke, Nakadai Masakazu, YAGUCHI Toshiaki, May 4, 2006: WO/2006/046593 (45 worldwide citation)

(EN) Disclosed is an excellent LXR modulator. Specifically disclosed is a compound represented by the general formula (I) below or the like. (I) [In the formula, R1 represents a -COR9 (wherein R9 represents an alkyl, optionally substituted alkoxy or optionally substituted amino); R2 represents an H, ...


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ASHWELL Mark A, KIZER Darin, MURAI Takahiro, NAKAI Daisuke, YASUKOCHI Takanori: COMPOSITIONS DE PYRROLOQUINOLÉINYL-PYRROLIDINE-2,5-DIONE ET PROCÉDÉS POUR PRÉPARER ET UTILISER CEUX-CI, PYRROLOQUINOLINYL-PYRROLIDINE-2,5-DIONE COMPOSITIONS AND METHODS FOR PREPARING AND USING SAME. ARQULE, ASHWELL Mark A, KIZER Darin, MURAI Takahiro, NAKAI Daisuke, YASUKOCHI Takanori, ELRIFI Ivor R, June 28, 2012: WO/2012/088491

The present invention relates to pyrroloquinolinyl-pyrrolidine-2,5-dione compounds and methods of synthesizing these compounds. The present invention also relates to pharmaceutical compositions containing pyrroloquinolinyl-pyrrolidine-2,5-dione compounds and methods of treating cell proliferative di ...