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Nicolae S Bodor, Kenneth B Sloan, Anwar A Hussain: Novel, transient pro-drug forms of L-DOPA to treat Parkinsons disease. Interx Research Corporation, Charles N Blitzer, July 12, 1977: US04035507 (82 worldwide citation)

There is provided, novel, transient pro-drug forms of L-DOPA (3,4-dihydroxy-L-phenylalanine), having the formula: ##STR1## wherein R represents a hydrogen atom, an acyl group, ##STR2## group, a -CO-pyridyl group, and a -CO-R.sub.3 group, wherein R.sub.3 represents the residue of any N,N-C.sub.1 -C.s ...


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Nicolae S Bodor, Kenneth B Sloan: Treating psoriasis with transient pro-drug forms of xanthine derivatives. INTERx Research Corporation, Charles N Blitzer, December 6, 1977: US04061753 (54 worldwide citation)

Compounds of the formula: ##STR1## wherein R, which may be the same or different, represents a member selected from the group consisting of --CH.sub.3, --C.sub.2 H.sub.5, --C.sub.3 H.sub.7, iso--C.sub.3 H.sub.7, --C.sub.4 H.sub.9, iso--C.sub.4 H.sub.9, pentyl, benzyl, allyl, 2-hydroxyethyl, cyclohex ...


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Nicolae S Bodor, Sun Shine Yuan: Intermediates useful in the synthesis of optically active m-acyloxy-.alpha.-[(methylamino)methyl]benzyl alcohols. Interx Research Corporation, Bacon & Thomas, June 12, 1979: US04158005 (51 worldwide citation)

Optically and therapeutically active compounds of the formula: ##STR1## wherein R represents a member selected from the group consisting of a straight or branched alkyl group of from one to twenty carbon atoms (C.sub.1 -C.sub.5 being preferred), an ethoxycarbonyl group, a benzyloxycarbonyl group, a ...


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Nicholas S Bodor, Kenneth B Sloan: Esteramide prodrugs of anti-inflammatory corticosteroids. INTERx Research Corporation, Burns Doane Swecker & Mathis, September 9, 1980: US04221787 (38 worldwide citation)

Transient, C-21 and/or C-17 esteramide prodrugs of the anti-inflammatory corticosteroids, prepared by esterification of hydroxy steroids, are disclosed.


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Nicolae S Bodor, Kenneth B Sloan, Anwar A Hussain: Novel, transient pro-drug forms of L-DOPA. Interx Research Corporation, Charles N Blitzer, December 21, 1976: US03998799 (32 worldwide citation)

There is provided, novel, transient pro-drug forms of L-DOPA (3,4-dihydroxy-L-phenylalanine), having the formula: ##STR1## wherein n represents an integer of from 2 to 50 with respect to formula (V-A), and wherein n represents an integer of from 1 to 50 with respect to formula (V-B);


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James J Kaminski, Nicolae S Bodor: 3-Chloro-2-oxazolidinones. Interx Research Corporation, Charles N Blitzer, January 6, 1976: US03931213 (27 worldwide citation)

Antibacterially effective 3-chloro-2-oxazolidinones are prepared by chlorination of an appropriate 2-oxazolidinone either with elemental chlorine in an aqueous medium or with a mono-, di- or trichloroisocyanuric acid (cyanuric chloride) in an inert organic solvent. The 2-oxazolidinones are, in turn, ...


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Kenji Nishimura, Mikio Arai, Kunihiro Sasahara, Takashi Nitanai: Effervescent enteric coated L-dopa formulation and method of using the same. Interx Research Corporation, Charles N Blitzer, June 1, 1976: US03961041 (26 worldwide citation)

Therapeutic levels of L-DOPA are achieved by orally administering a pharmaceutical effervescent-enteric coated tablet comprising:


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Valentino J Stella, Kenneth B Sloan: 5,5-Diphenylhydantoins. INTERx Research Corporation, Burns Doane Swecker & Mathis, April 7, 1981: US04260769 (25 worldwide citation)

Novel 5,5-diphenylhydantoins useful as anticonvulsants, antiepileptics and antiarrhythmics have the structural formula: ##STR1## wherein each R is hydrogen or --CH(R.sub.1)--X--P(O)(OH).sub.2, R.sub.1 is hydrogen or C.sub.1 -C.sub.7 straight or branched chain alkyl, and X is O or S, with the proviso ...


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Nicolae S Bodor: Labile, non-heterocyclic quaternary ammonium salt/esters as transient derivatives. Interx Research Corporation, Bacon & Thomas, July 3, 1979: US04160099 (25 worldwide citation)

Labile quaternary ammonium salts of the following formula (I) and (II) are provided: ##STR1## wherein ##STR2## represents a tertiary aliphatic amine; wherein ##STR3## represents an unsaturated amine; wherein R represents a member selected from the group consisting of a hydrogen atom, a C.sub.1 -C.su ...