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Hartmut Schirok, Joachim Mittendorf, Johannes Peter Stasch, Frank Wunder, Friederike Stoll, Karl Heinz Schlemmer: Pyrazolopyridine, indazole, imidazopyridine, imidazopyrimidine, pyrazolopyrazine and pyrazolopyridine derivatives as stimulators of guanylate cyclase for cardiovascular disorders. Bayer Intellectual Property, Karen B King, November 13, 2012: US08309551 (19 worldwide citation)

The present application relates to novel azabicyclic compounds, processes for their preparation, their use alone or in combinations for the treatment and/or prevention of diseases, and their use for producing medicaments for the treatment and/or prevention of diseases, especially for the treatment a ...


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Adrian Funke, Torsten Wagner, Ralph Lipp: Stabilised supersaturated solids of lipophilic drugs. Bayer Intellectual Property, Millen White Zelano Branigan P C, May 6, 2014: US08715735 (15 worldwide citation)

Methods for improving solubility and bioavailability of lipophilic compounds are described. Particularly, described are stabilized supersaturated solid solutions, particularly in power from, of lipophilic drugs, such as steroidal molecules.


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Markus Follmann, Johannes Peter Stasch, Gorden Redlich, Jens Ackerstaff, Nils Griebenow, Walter Kroh, Andreas Knorr, Eva Maria Becker, Frank Wunder, Volkhart Min Jian Li, Elke Hartmann, Joachim Mittendorf, Karl Heinz Schlemmer, Rolf Jautelat, Donald Bierer: Substituted 5-fluoro-1H-pyrazolopyridines and their use. Bayer Intellectual Property, Karen B King, April 16, 2013: US08420656 (15 worldwide citation)

The present application relates to novel substituted 5-fluoro-1H-pyrazolopyridines, to processes for their preparation, to their use alone or in combinations for the treatment and/or prophylaxis of diseases, and to their use for producing medicaments for the treatment and/or prophylaxis of diseases, ...


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FOLLMANN Markus, STASCH Johannes Peter, REDLICH Gorden, GRIEBENOW Nils, WUNDER Frank, LI Volkhart Min Jian, LANG Dieter: PYRAZOLOPYRIDINES SUBSTITUÉES PAR UN FLUORO-ALKYLE ET LEUR UTILISATION, FLUOROALKYL-SUBSTITUTED PYRAZOLOPYRIDINES AND USE THEREOF, FLUORALKYL-SUBSTITUIERTE PYRAZOLOPYRIDINE UND IHRE VERWENDUNG. BAYER INTELLECTUAL PROPERTY, FOLLMANN Markus, STASCH Johannes Peter, REDLICH Gorden, GRIEBENOW Nils, WUNDER Frank, LI Volkhart Min Jian, LANG Dieter, October 26, 2012: WO/2012/143510 (13 worldwide citation)

Die vorliegende Anmeldung betrifft neue Fluoralkyl-substituierte Pyrazolopyridine, Verfahren zu ihrer Herstellung, ihre Verwendung allein oder in Kombinationen zur Behandlung und/oder Prophylaxe von Krankheiten sowie ihre Verwendung zur Herstellung von Arzneimitteln zur Behandlung und/oder Prophylax ...


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HOFFMANN Sebastian, WASNAIRE Pierre, WACHENDORFF NEUMANN Ulrike: COMBINAISONS DE COMPOSÉS ACTIFS, ACTIVE COMPOUND COMBINATIONS. BAYER INTELLECTUAL PROPERTY, HOFFMANN Sebastian, WASNAIRE Pierre, WACHENDORFF NEUMANN Ulrike, December 13, 2012: WO/2012/168188 (13 worldwide citation)

The present invention relates to active compound combinations, in particular within a fungicide composition, which comprises (A) a thiazolylisoxazoline of formula (I) and a further fungicidally active compound (B). Moreover, the invention relates to a method for curatively or preventively controllin ...


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EIS Knut, PÜHLER Florian, ZORN Ludwig, SCHOLZ Arne, LIENAU Philip, GNOTH Mark Jean, BÖMER Ulf, GÜNTHER Judith, FANGHÄNEL Jörg, KORR Daniel: HÉTÉROCYCLYLAMINOIMIDAZOPYRIDAZINES, HETEROCYCLYL AMINOIMIDAZOPYRIDAZINES. Bayer Intellectual Property, EIS Knut, PÜHLER Florian, ZORN Ludwig, SCHOLZ Arne, LIENAU Philip, GNOTH Mark Jean, BÖMER Ulf, GÜNTHER Judith, FANGHÄNEL Jörg, KORR Daniel, BAYER INTELLECTUAL PROPERTY, December 27, 2012: WO/2012/175591 (10 worldwide citation)

The present invention relates to heterocyclyl aminoimidazopyridazine compounds of general formula (I) : in which A, R1, R2, R3 and R4 are as defined in the claims, to methods of preparing said compounds, to pharmaceutical compositions and combinations comprising said compounds and to the use of said ...


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FLAMME INGO, ERGUEDEN JENS KERIM, OEHME FELIX, THEDE KAI, KARIG GUNTER, KUHL ALEXANDER, WILD HANNO, SCHUHMACHER JOACHIM, KOLKHOF PETER, BAERFACKER LARS, HUETTER JOACHIM: DIPYRIDYL-DIHYDROPYRAZOLONES ET LEUR UTILISATION, DIPYRIDYL-DIHYDROPYRAZOLONES AND THEIR USE. BAYER HEALTHCARE, BAYER INTELLECTUAL PROPERTY, FETHERSTONHAUGH & CO, October 1, 2013: CA2608099 (9 worldwide citation)

The present application relates to novel dipyridyl-dihydropyrazolones, processes for their preparation, their use for treatment and/or prophylaxis of diseases and their use for the preparation of medicaments for treatment and/or prophylaxis of diseases, in particular cardiovascular and hematological ...


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KNUT Eis, PÜHLER Florian, ZORN Ludwig, SCHOLZ Arne, LIENAU Philip, GNOTH Mark, BÖMER Ulf, GÜNTHER Judith, FANGHÄNEL Jörg, KORR Daniel: AMINOIMIDAZOPYRIDAZINES SUBSTITUÉES, SUBSTITUTED AMINOIMIDAZOPYRIDAZINES. BAYER INTELLECTUAL PROPERTY, KNUT Eis, PÜHLER Florian, ZORN Ludwig, SCHOLZ Arne, LIENAU Philip, GNOTH Mark, BÖMER Ulf, GÜNTHER Judith, FANGHÄNEL Jörg, KORR Daniel, December 6, 2012: WO/2012/163942 (9 worldwide citation)

The present invention relates to substituted aminoimidazopyridazine compounds of general formula (I) : in which A, R1, R2, R3 and R4 are as defined in the claims, to methods of preparing said compounds, to pharmaceutical compositions and combinations comprising said compounds and to the use of said ...