WO/2011/034907 is referenced by 50 patents.

The invention relates to protein conjugates that contain a protein kinase containgn a cysteine residue in the ATP binding site and an inhibitor that is covalently and irreversibly bonded to said cysteine residue, such that the activity of the protein kinase is irreversibly inhibited. The invention also relates to compounds that irreversibly inhibit protein kinases.

Title
Protein kinase conjugates and inhibitors
Application Number
PCT/US/2010/048916
Publication Number
2011/034907
Application Date
September 15, 2010
Publication Date
March 24, 2011
Inventor
SINGH JUSWINDER
Agent
Underwood Robert H
Assignee
AVILA THERAPEUTICS
IPC
C12N 09/12
A61K 31/519
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