06316482 is referenced by 27 patents and cites 2 patents.

This invention relates to new benzamide derivatives having a vasopressin antagonistic activity, etc. and represented by general formula (I):

wherein

R

1

is aryl optionally substituted with lower alkoxy, etc.,

R

2

is lower alkyl, etc.,

R

3

is hydrogen, etc.,

A is NH, etc.,

E is

etc.,

X is —CH═CH—, —CH═N—, or S, and

Y is a condensed heterocyclic group, etc.,

and pharmaceutically acceptable salts thereof, to processes for preparation thereof and to a pharmaceutical composition comprising the same.

Title
Benzamide derivatives having a vasopressin antagonistic activity
Application Number
9/614132
Publication Number
6316482 (B1)
Application Date
July 11, 2000
Publication Date
November 13, 2001
Inventor
Teruo Oku
Takatsuki
US
Yuki Sawada
Ushiku
US
Hitoshi Sawada
Tsukuba
US
Tatsuya Zenkoh
Kitasouma-gun
US
Takehiko Ohkawa
Yuki-gun
US
Hiroyuki Setoi
Tsukuba
US
Agent
Oblon Spivak McClelland Maier & Neustadt P C
US
Assignee
Fujisawa Pharmaceutical
US
IPC
A61K 31/415
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