05606048 is referenced by 68 patents and cites 22 patents.

A stereoselective glycosylation process for preparing beta- and alpha-anomer enriched 2'-deoxy-2',2'-difluoronucleosides and 2'-deoxy-2'-fluoronucleosides by reacting a concentrated alpha- or beta-anomer enriched 2 -deoxy-2,2-difluorocarbohydrate or 2-deoxy-2 -fluorocarbohydrate with at least a molar equivalent of a nucleobase derivative in a high boiling inert solvent.

Title
Stereoselective glycosylation process for preparing 2-Deoxy-2, 2-difluoronucleosides and 2-deoxy-2-fluoronucleosides
Application Number
902302
Publication Number
5606048
Application Date
November 17, 1994
Publication Date
February 25, 1997
Inventor
Douglas P Kjell
West Lafayette
IN, US
Laurie M Poteet
Zionsville
IN, US
Ta Sen Chou
Indianapolis
IN, US
Agent
David E Boone
Joseph A Jones
Margaret M Brumm
Assignee
Eli Lilly and Company
IN, US
IPC
C07H 19/00
C07H 1/00
View Original Source