05426183 is referenced by 85 patents and cites 15 patents.

A catalytic stereoselective glycosylation process for preparing beta- and alpha-anomer enriched 2'-deoxy-2',2'-difluoronucleosides and 2'-deoxy-2'-fluoronucleosides involving reacting an alpha- or beta- anomer enriched 2-deoxy-2,2-difluorocarbohydrate or 2-deoxy-2-fluorocarbohydrate with at least a molar equivalent of a nucleobase derivative in an inert solvent and in the presence of a catalyst.

Title
Catalytic stereoselective glycosylation process for preparing 2-deoxy-2,2-difluoronucleosides and 2-deoxy-2-fluoronucleosides
Application Number
902112
Publication Number
5426183
Application Date
April 7, 1993
Publication Date
June 20, 1995
Inventor
Douglas P Kjell
West Lafayette
IN, US
Agent
David E Boone
Robert A Conrad
Assignee
Eli Lilly and Company
IN, US
IPC
C07D 405/04
View Original Source