05401838 is referenced by 50 patents and cites 14 patents.

A stereoselective fusion glycosylation process for prearing beta-anomer enriched 2'-deoxy-2',2'-difluoronucleotides and 2'-deoxy-2'-fluoronucleosides by reacting an alpha-anomer enriched 2-deoxy-2,2-difluorocarbohydrate or 2-deoxy-2-fluorcarbohydrate with at least a 3 molar equivalent of a nucleobase derivative at a temperature sufficient to melt the carbohydrate and nucleobase derivative.

Title
Stereoselective fusion glycosylation process for preparing 2-deoxy-2,2-difluoronucleosides and 2-deoxy-2-fluoronucleosides
Application Number
902312
Publication Number
5401838
Application Date
April 7, 1993
Publication Date
March 28, 1995
Inventor
Ta Sen Chou
Indianapolis
IN, US
Agent
David E Boone
Robert A Conrad
Sidney Persley
Assignee
Eli Lilly and Company
IN, US
IPC
C07H 19/19
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