0763524-A1 is referenced by 1 patents and cites 6 patents.

Compounds of formula (I): wherein: R is alkyl; R, R, R and R are the same or different and each is hydrogen, optionally substituted alkyl or various other organic groups; R is alkyl; R is a group of formula (II), (III), (IV), (V), (VI), (VII), (VIII) or (IX): wherein: A is a single bond, alkylene or alkenylene; A is or alkenylene; A is a single bond, alkyleneor alkenylene; R and R are the same or different and each is hydrogen, alkyl or various other groups; R is alkyl or phenyl; R is hydrogen or alkyl; R is alkyl or various other groups; and n is 0 or 1Ü and pharmaceutically acceptable salts thereof have valuable inhibitory activity against acyl-CoA: cholesterol acyl transferase.

Title
Urea and amide derivatives having acat inhibitory activity, their preparation and their therapeutic and prophylactic use
Application Number
EP19960306781 19960918
Publication Number
0763524 (A1)
Application Date
September 18, 1996
Publication Date
March 19, 1997
Inventor
Tokui Taro
JP
Kitazawa Eiichi
JP
Koga Teiichiro
JP
Ishihara Sadao
JP
Hayakawa Ichiro
JP
Kogen Hiroshi
JP
Shimada Kousei
JP
Kasai Takashi
JP
Oda Kozo
JP
Yoshida Akira
JP
Assignee
Sankyo Co
JP
IPC
C07C 311/32
C07C 311/29
C07C 311/04
C07C 275/42
C07C 275/40
C07C 275/38
C07C 275/34
C07C 275/32
C07C 275/24
C07C 271/64
C07C 271/20
C07C 271/12
C07C 259/10
C07C 255/60
C07C 255/57
C07C 255/49
C07C 255/44
C07C 255/01
C07C 251/48
C07C 237/52
C07C 237/42
C07C 237/22
C07C 235/38
C07C 233/08
A61P 09/10
A61K 31/535
A61K 31/445
A61K 31/40
A61K 31/275
A61K 31/18
A61K 31/17
A61K 31/16
C07C 275/28
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