0293881-A2 is referenced by 124 patents and cites 2 patents.

Peptides comprising C-terminal boronic acid derivatives of lysine, ornithine, and arginine, homoarginine and corresponding isothiouronium analogs thereof, of the formula are reversible inhibitors of trypsin-like serine proteases such as thrombin, plasma kallikrein and plasmin.

Title
Peptide boronic acid inhibitors of trypsin-like proteases.
Application Number
EP19880108817 19880601
Publication Number
0293881 (A2)
Application Date
June 1, 1988
Publication Date
December 7, 1988
Inventor
Shenvi Ashokkumar Bhikkappa
Kettner Charles Adrian
Assignee
Du Pont
US
IPC
C07K 05/00
C07F 05/02
A61K 37/64
A61K 31/69
C12N 09/99
C07K 14/81
C07K 05/00
C07F 05/00
A61P 29/00
A61P 07/00
A61K 38/55
C12N 09/99
C07K 14/81
C07K 05/10
C07K 05/08
C07K 05/06
C07K 05/00
C07F 05/02
A61P 29/00
A61P 07/02
A61K 38/55
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