0118364-A1 is referenced by 2 patents and cites 2 patents.

Compounds of the general formula: wherein R1, R2 and R3 are independently H or -@CH3; R4 is -@CH3 or an acoxycarbonyl group of the formula: -C@-O-R10 wherein R10 is C1-50 alkyl; 1- or 2-adamantyl; or 3-cholesteryl; R is H or C1-10 alkyl; provided that when R5 is C1-10 alkyl, the stereochemistry at chiral center I is either D or L; R6 is H or R6-R7 together is -CH2-CH2-CH2-; R7 is H, C1-7 alkyl, hydroxymethyl, mercaptomethyl, benzyl or p-hydroxybenzyl; provided that when R7 is not H, the stereochemistry at chiral center II is L; R8 and R9 are independently -COOR or -CONR min R sec wherein R is H or C1-7 alkyl, and R min and R sec are independently H or C1-3 alkyl; the stereochemistry at chiral center III is always D. These compounds possess adjuvant and immunostimulatory properties.

Immunostimulatory dipeptidyl d-glucose derivatives and methods of preparation.
Application Number
EP19840400413 19840301
Publication Number
0118364 (A1)
Application Date
March 1, 1984
Publication Date
September 12, 1984
Shen T Y
Durette Philippe L
Dorn Conrad P
Merck & Co
A61K 39/39
A61K 31/70
C07H 15/00
C07K 09/00
C07K 01/00
A61P 37/00
A61K 39/39
A61K 38/00
C07K 09/00
C07K 01/113
A61P 37/00
A61K 39/39
A61K 38/00
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